A Base Promoted Cyclization of N-Propargylaminopyridines. Synthesis of Imidazo[1,2-a]pyridine Derivatives
Само за регистроване кориснике
2011
Чланак у часопису (Објављена верзија)
Метаподаци
Приказ свих података о документуАпстракт
A base promoted cyclization of the protected N-propargylaminopyridines was shown to be an efficient method for the preparation of imidazo[1,2-a] pyridine derivatives. The reactions were carried out with a small excess of base, at room temperature or slightly above producing the heterocyclic products in moderate to good yields. The stereoelectronic properties of substituents on the pyridine ring were shown to influence the cyclization process.
Извор:
Organic Letters, 2011, 13, 9, 2286-2289Издавач:
- Amer Chemical Soc, Washington
Финансирање / пројекти:
- Компјутерско дизајнирање, синтеза и биолошка евалуација нових хетероцикличних једињења као селективних инхибитора туморогенезе (RS-MESTD-Basic Research (BR or ON)-172009)
DOI: 10.1021/ol200508x
ISSN: 1523-7060
PubMed: 21446664
WoS: 000289956700037
Scopus: 2-s2.0-79955576570
Институција/група
PharmacyTY - JOUR AU - Husinec, Suren AU - Marković, Rade AU - Petković, Miloš AU - Nasufović, Veselin AU - Savić, Vladimir PY - 2011 UR - https://farfar.pharmacy.bg.ac.rs/handle/123456789/1527 AB - A base promoted cyclization of the protected N-propargylaminopyridines was shown to be an efficient method for the preparation of imidazo[1,2-a] pyridine derivatives. The reactions were carried out with a small excess of base, at room temperature or slightly above producing the heterocyclic products in moderate to good yields. The stereoelectronic properties of substituents on the pyridine ring were shown to influence the cyclization process. PB - Amer Chemical Soc, Washington T2 - Organic Letters T1 - A Base Promoted Cyclization of N-Propargylaminopyridines. Synthesis of Imidazo[1,2-a]pyridine Derivatives VL - 13 IS - 9 SP - 2286 EP - 2289 DO - 10.1021/ol200508x ER -
@article{ author = "Husinec, Suren and Marković, Rade and Petković, Miloš and Nasufović, Veselin and Savić, Vladimir", year = "2011", abstract = "A base promoted cyclization of the protected N-propargylaminopyridines was shown to be an efficient method for the preparation of imidazo[1,2-a] pyridine derivatives. The reactions were carried out with a small excess of base, at room temperature or slightly above producing the heterocyclic products in moderate to good yields. The stereoelectronic properties of substituents on the pyridine ring were shown to influence the cyclization process.", publisher = "Amer Chemical Soc, Washington", journal = "Organic Letters", title = "A Base Promoted Cyclization of N-Propargylaminopyridines. Synthesis of Imidazo[1,2-a]pyridine Derivatives", volume = "13", number = "9", pages = "2286-2289", doi = "10.1021/ol200508x" }
Husinec, S., Marković, R., Petković, M., Nasufović, V.,& Savić, V.. (2011). A Base Promoted Cyclization of N-Propargylaminopyridines. Synthesis of Imidazo[1,2-a]pyridine Derivatives. in Organic Letters Amer Chemical Soc, Washington., 13(9), 2286-2289. https://doi.org/10.1021/ol200508x
Husinec S, Marković R, Petković M, Nasufović V, Savić V. A Base Promoted Cyclization of N-Propargylaminopyridines. Synthesis of Imidazo[1,2-a]pyridine Derivatives. in Organic Letters. 2011;13(9):2286-2289. doi:10.1021/ol200508x .
Husinec, Suren, Marković, Rade, Petković, Miloš, Nasufović, Veselin, Savić, Vladimir, "A Base Promoted Cyclization of N-Propargylaminopyridines. Synthesis of Imidazo[1,2-a]pyridine Derivatives" in Organic Letters, 13, no. 9 (2011):2286-2289, https://doi.org/10.1021/ol200508x . .