Преглед аутора: "Cook, James M."
Приказ резултата 1-20 од 64
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Acute effects of an inverse agonist selective for alpha(5) GABA(A) receptors on rat behaviour in the forced swim test
Samardžić, Janko; Batinić, Bojan; Biawat, Poonam; Obradović, Dragan I.; Cook, James M.; Savić, Miroslav (Elsevier Science BV, Amsterdam, 2012) -
Are GABA(A) receptors containing alpha 5 Subunits contributing to the sedative properties of benzodiazepine site agonists?
Savić, Miroslav; Huang, Shengming; Furtmueller, Roman; Clayton, Terry; Huck, Sigismund; Obradović, Dragan I.; Ugrešić, Nenad; Sieghart, Werner; Bokonjić, Dubravko; Cook, James M. (Nature Publishing Group, London, 2008) -
Attaining in vivo selectivity of positive modulation of alpha 3 ss gamma 2 GABA(A) receptors in rats: A hard task!
Batinić, Bojan; Stanković, Tamara; Stephen, Michael; Kodali, Revathi; Tiruveedhula, Veera V.; Li, Guanguan; Scholze, Petra; Marković, Bojan; Obradović, Aleksandar; Ernst, Margot; Cook, James M.; Savić, Miroslav (Elsevier Science BV, Amsterdam, 2018) -
Attaining in vivo selectivity of positive modulation of GABAA ɑ3 receptors in rats: a hard task
Batinić, Bojan; Stanković, Tamara; Poe, Michael M.; Cook, James M.; Savić, Miroslav (Elsevier Science BV, Amsterdam, 2016) -
Behavioural Characterization of Four Endemic Stachys Taxa
Savić, Miroslav; Kukić-Marković, Jelena; Grayer, Renee J.; Milinković, Marija M.; Marin, Petar; Divljaković, Jovana; van Linn, Michael; Cook, James M.; Petrović, Silvana (Wiley-Blackwell, Malden, 2010) -
Benzodiazepine site inverse agonists and locomotor activity in rats: Bimodal and biphasic influence
Savić, Miroslav; Obradović, Dragan I.; Ugrešić, Nenad; Cook, James M.; Yin, Wenyuan; van Linn, Michael; Bokonjić, Dubravko (Pergamon-Elsevier Science Ltd, Oxford, 2006) -
Benzodiazepine-induced spatial learning deficits in rats are regulated by the degree of modulation of α 1 GABA A receptors
Joksimović, Srđan; Divljaković, Jovana; van Linn, Michael; Varagić, Zdravko; Brajković, Gordana; Milinković, Marija M.; Yin, Wenyuan; Timić, Tamara; Sieghart, Werner; Cook, James M.; Savić, Miroslav (European Neuropsychopharmacology, 2013) -
Beta CCT as well as flumazenil prevent the diazepam withdrawal-induced anxiety in the elevated plus maze in rats
Divljaković, Jovana; Timić, Tamara; Milinković, Marija M.; Batinić, Bojan; van Linn, Michael; Cook, James M.; Savić, Miroslav (Oxford Univ Press, Oxford, 2012) -
Biocompatible nanoemulsions as a tool for preclinical testing of CW-02-79, a pyrazoloquinolinone modulator of sigma-2 receptors: preformulation and formulation studies
Ilić, Tanja; Stanković, Tijana; Mitrović, Jelena; Pantelić, Ivana; Dobričić, Vladimir; Cook, James M.; Savić, Miroslav; Savić, Snežana (4th European Conference on Pharmaceutics, 20 - 21 March 2023, Marseille, France, 2023) -
Comparative anticonvulsant activity of the GABAkine KRM-II-81 and a deuterated analog
Ping, Xingjie; Meyer, Michelle J.; Zahn, Nicolas M.; Golani, Lalit K.; Sharmin, Dishary; Pandey, Kamal P.; Revanian, Sepideh; Mondal, Prithu; Jin, Xiaoming; Arnold, Leggy A.; Cerne, Rok; Cook, James M.; Divović, Branka; Savić, Miroslav; Lippa, Arnold; Smith, Jodi L.; Witkin, Jeffrey M. (John Wiley and Sons Inc, 2023) -
Contribution of a1 subunit-containing GABA-A receptors to diazepam-induced motor impairment
Divljaković, Jovana; van Linn, Michael; Milinković, Marija M.; Yin, Wenyuan; Batinić, Bojan; Cook, James M.; Savić, Miroslav (Elsevier Science BV, Amsterdam, 2010) -
Design and synthesis of novel deuterated GABAAR-alpha 6 subtype selective ligands with improved metabolic stability and enhanced bioavailability
Knutson, Daniel; Kodali, Revathi; Stephen, Michael; Verma, Ranjit; Witzigmann, Christopher; Meirelles, Matheus; Zahn, Nicolas; Huber, Alec; Arnold, Leggy; Savić, Miroslav; Ernst, Margot; Sieghart, Werner; Cook, James M. (Amer Chemical Soc, Washington, 2018) -
Design and Synthesis of Novel Deuterated Ligands Functionally Selective for the gamma-Aminobutyric Acid Type A Receptor (GABA(A)R) alpha 6 Subtype with Improved Metabolic Stability and Enhanced Bioavailability
Knutson, Daniel; Kodali, Revathi; Divović, Branka; Treven, Marco; Stephen, Michael; Zahn, Nicolas; Dobričić, Vladimir; Huber, Alec; Meirelles, Matheus; Verma, Ranjit; Wimmer, Laurin; Witzigmann, Christopher; Arnold, Leggy; Chiou, Lih-Chu; Ernst, Margot; Mihovilović, Marko D.; Savić, Miroslav; Sieghart, Werner; Cook, James M. (Amer Chemical Soc, Washington, 2018) -
Design and synthesis of stereoenantiomeric benzodiazepine receptor ligands
Huang, Shengming; Savić, Miroslav; Furtmueller, Roman; Duke, Angela; Clayton, Terry; Sieghart, Werner; Rowlett, James K.; Cook, James M. (Amer Chemical Soc, Washington, 2007) -
Design of tailor-made biocompatible nanocarrier for novel pyrazoloquinolinone ligand (CW-02-79) based on comprehensive evaluation of critical physicochemical descriptors
Stanković, Tijana; Ilić, Tanja; Pantelić, Ivana; Tošić, Anđela; Mitrović, Jelena; Cook, James M.; Savić, Miroslav; Savić, Snežana (International Association of Physical Chemists, 2023) -
The differential role of alpha(1)- and alpha(5)-containing GABA(A) receptors in mediating diazepam effects on spontaneous locomotor activity and water-maze learning and memory in rats
Savić, Miroslav; Milinković, Marija M.; Rallapalli, Sundari; Clayton, Terry; Joksimović, Srđan; van Linn, Michael; Cook, James M. (Oxford Univ Press, Oxford, 2009) -
Duration of treatment and activation of alpha(1)-containing GABA(A) receptors variably affect the level of anxiety and seizure susceptibility after diazepam withdrawal in rats
Kovacević, Jovana; Timić, Tamara; Tiruveedhula, Veera V.; Batinić, Bojan; Namjoshi, Ojas A.; Milić, Marija; Joksimović, Srđan; Cook, James M.; Savić, Miroslav (Pergamon-Elsevier Science Ltd, Oxford, 2014) -
Effects of a novel inverse agonist selective for alpha5 GABAA receptors on spatial memory: comparison with the standard non-selective inverse agonist DMCM
Samardžić, Janko; Savić, Miroslav; Clayton, Terry; Rallapalli, Sundari; Obradović, Dragan I.; Joksimović, Srđan; Sieghart, Werner; Cook, James M. (Elsevier Science BV, Amsterdam, 2008) -
Effects of positive alpha5-selective modulation of GABA A receptors on amphetamine-induced hyperlocomotion
Timić-Stamenić, Tamara; Santrač, Anja; Divović, Branka; Poe, Michael M.; Cook, James M.; Savić, Miroslav (Elsevier Science BV, Amsterdam, 2015) -
Effects of PWZ-029, an alpha(5)GABA(A) receptor inverse agonist, on scopolamine-induced spatial learning deficits in the water maze
Joksimović, Srđan; Timić, Tamara; Radulović, Tamara; Rallapalli, Sundari; Milinković, Marija M.; Divljaković, Jovana; Batinić, Bojan; Cook, James M.; Savić, Miroslav (Elsevier Science BV, Amsterdam, 2012)