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Data mining implementation in multiparticulate unit systems characterization
(Macedonian Pharmaceutical AssociationSs. Cyril and Methodius University in Skopje, Faculty of Pharmacy, 2023)
Multiparticulate unit systems (MPUs) represent
versatile drug delivery systems which provide flexible
dosing and reproducible drug release profile (Al-Hashimi
et al., 2018). They are usually filled in capsules/sachets ...
Applicability of Expert System for Drug Development as a tool for co-processed excipients formulation development
(Macedonian Pharmaceutical AssociationFaculty of Pharmacy, Ss Cyril and Methodius University in Skopje, 2022)
Expert System for Drug Development, i.e. SeDeM
Expert System (Span. Sistema Experto para DEsarrollo
de Medicamentos) represents a method intended for
evaluation of powder properties affecting processability,
particularly ...
Preformulation and development of preliminary nanoemulsion carrier for patent protected compound GL-II-73
(Macedonian Pharmaceutical AssociationSs. Cyril and Methodius University in Skopje, Faculty of Pharmacy, 2023)
Nanopharmaceuticals offer a good option to avoid
some of the difficulties that novel drug candidates
confront. They can be tailored to adjust their water
solubility, half-life, biodistribution, and govern the release
of ...
Anatomical characterization, chemical analyses and essential oil antimicrobial activity of Hyssopus officinalis L. (Lamiaceae)
(Macedonian Pharmaceutical AssociationSs. Cyril and Methodius University in Skopje, Faculty of Pharmacy, 2022)
Introduction
Hyssopus officinalis L. (Lamiaceae) is a perennial aromatic subshrub, distributed mainly in the Mediterranean area. The aerial parts of the plant are used as a culinary and medicinal herb (Hyssopi herba) ...
In silico assessment of intestinal precipitation: Case study of a poorly soluble, weakly basic compound
(Macedonian Pharmaceutical AssociationSs. Cyril and Methodius University in Skopje, Faculty of Pharmacy, 2023)
Precipitation of a drug substance in the small intestine
is a phenomenon relevant to weak bases due to their pH-
dependent solubility. Because of the low solubility at
higher pH, upon entry in the small intestine, a ...
Selenium nanoparticles render pandrug-resistant Acinetobacter baumannii susceptible to colistin
(Macedonian Pharmaceutical Association, 2022)
Colistin is used as a “last resort” drug in the treatment
of carbapenem-resistant Acinetobacter baumannii
infections. Though not the most convenient option due to
the serious side effects, this antibiotic can be very ...
Pharmaceutical and technological characteristics of barium sulphate tablets -the screening of various formulation factors
(Macedonian Pharmaceutical AssociationFaculty of Pharmacy, Ss Cyril and Methodius University in Skopje, 2022)
Introduction The study examined the development of barium sulphate tablets that do not dissolve in the digestive tract
and are used as a contrasting agent for measuring transit time through the column. The main problem ...
Characterization of chitosan/xanthan gum polyelectrolyte complexes as carriers for ibuprofen: influence of drug encapsulation procedure on complex formation
(Macedonian Pharmaceutical AssociationFaculty of Pharmacy, Ss Cyril and Methodius University in Skopje, 2020)
Introduction
Ibuprofen (IBU) is commonly used non-steroidal
anti-inflammatory drug. It is a weak acid (pKa ~4.5)
with low pH dependent aqueous solubility (46
μg/mL at pH 1.5 and ˃300 μg/mL at pH˃7, at 25
°C). The most ...
Fun-shaped oral dosage forms for the pediatric population fabricated by digital light processing (DLP) 3D printing technique
(Macedonian Pharmaceutical AssociationFaculty of Pharmacy, Ss Cyril and Methodius University in Skopje, 2022)
Introduction Three-dimensional (3D) printing as an innovative technology in the field of drug manufacturing has attracted a lot of attention from the scientific and professional public in recent years. Classified into seven ...
An investigation into applicability of sodium carboxymethylcellulose and sodium alginate as film-forming agents for semi-solid 3D printing
(Macedonian Pharmaceutical AssociationSs. Cyril and Methodius University in Skopje, Faculty of Pharmacy, 2023)
Semi-solid 3D printing technology has gained
increased interest in the pharmaceutical field as it enables
on-demand fabrication of personalized dosage forms.
Orodispersible films (ODFs) are good candidates for 3D
printing ...