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Adverse effects and toxicity of analgesics

Neželjeni efekti i toksičnost analgetika

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2012
1782.pdf (266.1Kb)
Authors
Bulat, Zorica
Matović, Vesna
Article (Published version)
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Abstract
Even though among the most widely used analgoantipiretics with confirmed pharmacological effects, acetylsalicylic acid, paracetamol and ibuprofen may be the cause of poisonings and even death. Acetylsalicylic acid and paracetamol are most commonly used drugs that are dispensed without a prescription. However, poison control centers are warning of the risk associated with the use of these COX inhibitors. It is well known that acetylsalicylic acid causes prolonged inhibition of blood coagulation, metabolic acidosis and other toxic effects while the toxic effects of paracetamol are mainly manifested on liver. Ibuprofen poisoning is much rarer, especially those leading to death. Ibuprofen overdose can cause mainly gastrointestinal disturbances, and can also lead to renal damage.
U ovom radu obrađeni su acetilsalicilna kiselina, paracetamol i ibuprofen, s obzirom da su među najšire korišćenim analgoantipireticima koji i pored neosporno potvrđenog farmakološkog dejstva mogu biti uzročnici trovanja, pa i smrti. Acetilsalicilna kiselina i paracetamol su najčešće korišćeni lekovi koji se izdaju bez recepta, a izveštaji centara za kontrolu trovanja opominju na rizik koji nose ovi COX inhibitori. Poznato je da acetilsalicilna kiselina dovodi do produžene inhibicije koagulacije krvi, metaboličke acidoze i drugih toksičnih efekata, a da se toksičnost paracetamola prvenstveno ispoljava na jetri. Trovanja ibuprofenom su znatno ređa, posebno sa smrtnim ishodom. Pri predoziranju ibuprofenom dominiraju gastrointestinalne smetnje, a može doći i do renalnog oštećenja.
Keywords:
paracetamol / acetylsalicylic acid / ibuprofen / drug toxicity / poisoning / paracetamol / acetilsalicilna kiselina / ibuprofen / toksičnost lekova / trovanja
Source:
Arhiv za farmaciju, 2012, 62, 2, 92-100
Publisher:
  • Savez farmaceutskih udruženja Srbije, Beograd
Funding / projects:
  • Improvement and development of hygienic and technological procedures in production of animal originating foodstuffs with the aim of producing high-quality and safe products competetive on the global market (RS-46009)

ISSN: 0004-1963

Scopus: 2-s2.0-84863789605
[ Google Scholar ]
Handle
https://hdl.handle.net/21.15107/rcub_farfar_1784
URI
https://farfar.pharmacy.bg.ac.rs/handle/123456789/1784
Collections
  • Radovi istraživača / Researchers’ publications
Institution/Community
Pharmacy
TY  - JOUR
AU  - Bulat, Zorica
AU  - Matović, Vesna
PY  - 2012
UR  - https://farfar.pharmacy.bg.ac.rs/handle/123456789/1784
AB  - Even though among the most widely used analgoantipiretics with confirmed pharmacological effects, acetylsalicylic acid, paracetamol and ibuprofen may be the cause of poisonings and even death. Acetylsalicylic acid and paracetamol are most commonly used drugs that are dispensed without a prescription. However, poison control centers are warning of the risk associated with the use of these COX inhibitors. It is well known that acetylsalicylic acid causes prolonged inhibition of blood coagulation, metabolic acidosis and other toxic effects while the toxic effects of paracetamol are mainly manifested on liver. Ibuprofen poisoning is much rarer, especially those leading to death. Ibuprofen overdose can cause mainly gastrointestinal disturbances, and can also lead to renal damage.
AB  - U ovom radu obrađeni su acetilsalicilna kiselina, paracetamol i ibuprofen, s obzirom da su među najšire korišćenim analgoantipireticima koji i pored neosporno potvrđenog farmakološkog dejstva mogu biti uzročnici trovanja, pa i smrti. Acetilsalicilna kiselina i paracetamol su najčešće korišćeni lekovi koji se izdaju bez recepta, a izveštaji centara za kontrolu trovanja opominju na rizik koji nose ovi COX inhibitori. Poznato je da acetilsalicilna kiselina dovodi do produžene inhibicije koagulacije krvi, metaboličke acidoze i drugih toksičnih efekata, a da se toksičnost paracetamola prvenstveno ispoljava na jetri. Trovanja ibuprofenom su znatno ređa, posebno sa smrtnim ishodom. Pri predoziranju ibuprofenom dominiraju gastrointestinalne smetnje, a može doći i do renalnog oštećenja.
PB  - Savez farmaceutskih udruženja Srbije, Beograd
T2  - Arhiv za farmaciju
T1  - Adverse effects and toxicity of analgesics
T1  - Neželjeni efekti i toksičnost analgetika
VL  - 62
IS  - 2
SP  - 92
EP  - 100
UR  - https://hdl.handle.net/21.15107/rcub_farfar_1784
ER  - 
@article{
author = "Bulat, Zorica and Matović, Vesna",
year = "2012",
abstract = "Even though among the most widely used analgoantipiretics with confirmed pharmacological effects, acetylsalicylic acid, paracetamol and ibuprofen may be the cause of poisonings and even death. Acetylsalicylic acid and paracetamol are most commonly used drugs that are dispensed without a prescription. However, poison control centers are warning of the risk associated with the use of these COX inhibitors. It is well known that acetylsalicylic acid causes prolonged inhibition of blood coagulation, metabolic acidosis and other toxic effects while the toxic effects of paracetamol are mainly manifested on liver. Ibuprofen poisoning is much rarer, especially those leading to death. Ibuprofen overdose can cause mainly gastrointestinal disturbances, and can also lead to renal damage., U ovom radu obrađeni su acetilsalicilna kiselina, paracetamol i ibuprofen, s obzirom da su među najšire korišćenim analgoantipireticima koji i pored neosporno potvrđenog farmakološkog dejstva mogu biti uzročnici trovanja, pa i smrti. Acetilsalicilna kiselina i paracetamol su najčešće korišćeni lekovi koji se izdaju bez recepta, a izveštaji centara za kontrolu trovanja opominju na rizik koji nose ovi COX inhibitori. Poznato je da acetilsalicilna kiselina dovodi do produžene inhibicije koagulacije krvi, metaboličke acidoze i drugih toksičnih efekata, a da se toksičnost paracetamola prvenstveno ispoljava na jetri. Trovanja ibuprofenom su znatno ređa, posebno sa smrtnim ishodom. Pri predoziranju ibuprofenom dominiraju gastrointestinalne smetnje, a može doći i do renalnog oštećenja.",
publisher = "Savez farmaceutskih udruženja Srbije, Beograd",
journal = "Arhiv za farmaciju",
title = "Adverse effects and toxicity of analgesics, Neželjeni efekti i toksičnost analgetika",
volume = "62",
number = "2",
pages = "92-100",
url = "https://hdl.handle.net/21.15107/rcub_farfar_1784"
}
Bulat, Z.,& Matović, V.. (2012). Adverse effects and toxicity of analgesics. in Arhiv za farmaciju
Savez farmaceutskih udruženja Srbije, Beograd., 62(2), 92-100.
https://hdl.handle.net/21.15107/rcub_farfar_1784
Bulat Z, Matović V. Adverse effects and toxicity of analgesics. in Arhiv za farmaciju. 2012;62(2):92-100.
https://hdl.handle.net/21.15107/rcub_farfar_1784 .
Bulat, Zorica, Matović, Vesna, "Adverse effects and toxicity of analgesics" in Arhiv za farmaciju, 62, no. 2 (2012):92-100,
https://hdl.handle.net/21.15107/rcub_farfar_1784 .

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