Приказ основних података о документу

dc.creatorGagić, Žarko
dc.creatorRužić, Dušan
dc.creatorĐoković, Nemanja
dc.creatorĐikić, Teodora
dc.creatorNikolić, Katarina
dc.date.accessioned2020-02-12T11:57:05Z
dc.date.available2020-02-12T11:57:05Z
dc.date.issued2020
dc.identifier.issn2296-2646
dc.identifier.urihttps://farfar.pharmacy.bg.ac.rs/handle/123456789/3502
dc.description.abstractRational drug design implies usage of molecular modeling techniques such as pharmacophore modeling, molecular dynamics, virtual screening, and molecular docking to explain the activity of biomolecules, define molecular determinants for interaction with the drug target, and design more efficient drug candidates. Kinases play an essential role in cell function and therefore are extensively studied targets in drug design and discovery. Kinase inhibitors are clinically very important and widely used antineoplastic drugs. In this review, computational methods used in rational drug design of kinase inhibitors are discussed and compared, considering some representative case studies.en
dc.publisherFrontiers Media S.A.
dc.relationinfo:eu-repo/grantAgreement/MESTD/Basic Research (BR or ON)/172033/RS//
dc.rightsopenAccess
dc.rights.urihttps://creativecommons.org/licenses/by/4.0/
dc.sourceFrontiers in Chemistry
dc.subjectdrug discovery
dc.subjectkinase inhibitors
dc.subjectmolecular modeling
dc.subjectpharmacophore
dc.subjectrational drug design
dc.titleIn silico Methods for Design of Kinase Inhibitors as Anticancer Drugsen
dc.typearticle
dc.rights.licenseBY
dcterms.abstractЂикић, Теодора; Николић, Катарина; Гагић, Жарко; Ружић, Душан; Ђоковић, Немања; Ин силицо Метходс фор Десигн оф Кинасе Инхибиторс ас Aнтицанцер Другс;
dc.citation.volume7
dc.citation.rankM21
dc.identifier.wos000615281300001
dc.identifier.doi10.3389/fchem.2019.00873
dc.identifier.scopus2-s2.0-85078245053
dc.identifier.fulltexthttps://farfar.pharmacy.bg.ac.rs/bitstream/id/7486/In_silico_Method_pub_2020.pdf
dc.type.versionpublishedVersion


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