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Pharmacological characterisation of Seseli gracile Waldst. & Kit. (Apiaceae) essential oil
Farmakološka karakterizacija etarskog ulja Seseli gracile Waldst. & Kit. (Apiaceae)
dc.creator | Suručić, Relja | |
dc.creator | Kundaković-Vasović, Tatjana | |
dc.creator | Marčetić, Mirjana | |
dc.creator | Drakul, Dragana | |
dc.creator | Milenković, Marina | |
dc.creator | Kovačević, Nada | |
dc.date.accessioned | 2021-12-07T14:06:28Z | |
dc.date.available | 2021-12-07T14:06:28Z | |
dc.date.issued | 2021 | |
dc.identifier.issn | 0042-8450 | |
dc.identifier.uri | https://farfar.pharmacy.bg.ac.rs/handle/123456789/4002 | |
dc.description.abstract | Phytochemical and pharmacological in-vestigations of essential oils isolated from plant species of the genus Seseli have been intensified recently. These plant species have long-term use in nutrition and traditional medicine in the treatment of various disorders. Volatile secondary metabolites of Seseli gracile Waldst. & Kit (Apiaceae) have not been pharma-cologically examined so far. The aim of the conducted research was to assess the antiradical, antimicrobial and spasmolytic ac-tivities of S. gracile essential oil isolated from the aerial parts of the plant. Methods. The antiradical activity was determined us-ing the 2,2-diphenyl-1-picrylhydrazyl (DPPH) radical scaveng-ing test, antimicrobial activity using broth microdilution meth-od with standard strains of Gram (+), Gram (-) bacteria and yeast, while spasmolytic activity was evaluated on isolated rat il-eum, pre-contracted with a high concentration of potassium. Results. The results showed moderate antiradical (SC50 = 78.60 μg/mL) and good spasmolytic activity (IC50 = 271.4 nL/mL) of S. gracile essential oil. In the range of tested concen-trations, minimal inhibitory concentration (MIC) was deter-mined only for the strain of Escherichia coli (500 μg/mL). Con-clusion. Results obtained in this study justify the need for fur-ther studies to elucidate exact molecular mechanism underlay this spasmolytic effect of S. gracile herb essential oil. | |
dc.description.abstract | Etarska ulja izolovana iz vrsta roda Seseli su u poslednje vreme intenzivno farmakološki i fitohemijski proučavana. Biljke iz ovog roda se koriste već duži niz godina u ishrani i tradicionalnoj terapiji različitih oboljenja. Farmakološka aktivnost etarskog ulja izolovanog iz Seseli gracile do sada nije ispitivana. Stoga je cilj ovog istraživanja bio da se ispita antiradikalska, antimikrobna i spazmolitična aktivnost etarskog ulja izolovanog iz nadzemnih delova biljne vrste S. gracile. Metode. Antiradikalska aktivnost je utvrđena testom neutralizacije 2.2-difenil-1-pikrilhidrazil (DPPH) radikala, antimikrobna, bujon-mikrodilucionom metodom uz upotrebu standardnih sojeva Gram (+), Gram (-) bakterija i gljivica, a spazmolitična na izolovanom ileumu pacova, prethodno kontrahovanom visokom koncentarcijom kalijuma. Rezultati. Rezultati pokazuju umerenu antiradikalsku (SC50 = 78.60 μg/mL) i dobru spazmolitičnu aktivnost (IC50 = 271.4 nL/mL) etarskog ulja S. gracile. U opsegu testiranih koncentracija utvrđena je minimalna inhibitorna koncentracija (MIC) samo za soj Escherichia coli (500 μg/mL). Zaključak. Dobijeni rezultati opravdavaju potrebu za budućim istraživanjima koja bi razjasnila tačne mehanizme kojima se ostvaruje spazmolitički efekat etarskog ulja nadzemnog dela S. gracile. | |
dc.publisher | Belgrade : Military Medical Academy, INI | |
dc.relation | info:eu-repo/grantAgreement/MESTD/Basic Research (BR or ON)/173021/RS// | |
dc.rights | openAccess | |
dc.rights.uri | https://creativecommons.org/licenses/by-sa/4.0/ | |
dc.source | Vojnosanitetski pregled | |
dc.subject | Apiaceae | |
dc.subject | Antioxidants | |
dc.subject | Anti-infective agents | |
dc.subject | Muscle relaxation | |
dc.subject | Oils | |
dc.subject | Pharmacology | |
dc.subject | Plant extracts | |
dc.subject | Volatile | |
dc.subject | apiaceae | |
dc.subject | etarsko ulje | |
dc.subject | farmakologija | |
dc.subject | ekstrakti | |
dc.subject | biljni | |
dc.subject | mišić | |
dc.subject | relaksacija | |
dc.subject | antioksidanti | |
dc.subject | antiinfektivni agensi | |
dc.title | Pharmacological characterisation of Seseli gracile Waldst. & Kit. (Apiaceae) essential oil | |
dc.title | Farmakološka karakterizacija etarskog ulja Seseli gracile Waldst. & Kit. (Apiaceae) | |
dc.type | article | |
dc.rights.license | BY-SA | |
dc.citation.volume | 78 | |
dc.citation.issue | 10 | |
dc.citation.spage | 1065 | |
dc.citation.epage | 1071 | |
dc.citation.rank | M23 | |
dc.identifier.wos | 000715905000007 | |
dc.identifier.doi | 10.2298/VSP190320028S | |
dc.identifier.scopus | 2-s2.0-85119899899 | |
dc.identifier.fulltext | http://farfar.pharmacy.bg.ac.rs/bitstream/id/9313/Pharmacological_characterisation_of_pub_2021.pdf | |
dc.type.version | publishedVersion |