Preparations of laxatives and antidiarrhoeals: Pharmaceutically - technological aspect
Lekoviti preparati lakasativa i antidijaroika - farmaceutsko tehnološki aspekt
Abstract
In this report preparations of laxatives and antidiarrhoeals and the technological procedures used in production, have been reviewed.The importance of special technological procedure as freeze drying in the production and stabilisation has been explained. The most frequent dosage forms for these drugs are tablets.Good physical characteristics of tablets, insignificant variation of drug content, uniformity of dosage as required bioavailability are to bi provided by using adequate combination of excipients in the formulation and by proper selection of production method and order of technological operations.Additional requirements are to be achieved in the production of chewable tablets , frequently used as a dosage form for laxatives as calcium polycarbophil. Basic concept of tablet production validation is included in this report.
U radu su prikazani lekoviti preparati laksativa i antidijaroika i metode koje se koriste u proizvodnji. Objašnjen je značaj specijalnih tehnoloških postupaka kao što je liofilizacija u proizvodnji i stabilizaciji nekih proizvoda iz ove grupe.Najčešće primenjivani oblik ovih lekovitih supstanci su tablete. Za proizvodnju tableta koje će imati dobre fizičke karakteristike, zanemarljivo mala odstupanja u sadržaju leka, jednolikost doze kao i potrebnu bioraspoloživost, koristi se adekvatna kombinacija pomoćnih materija u formulaciji i pravilan izbor metode izrade. Dodatni zahtevi se postavljaju u slučaju proizvodnje tableta za žvakanje, kao što su tablete sa kalcijum polikarbofilom. U radu su dati i osnovni principi validacije procesa proizvodnje tableta.
Keywords:
laxatives / antidiarrhoeals / freeze drying / tablet production validation / laksativi / antidijaroici / sušenje smrzavanjem / validacija proizvodnje tabletaSource:
Arhiv za farmaciju, 2004, 54, 3, 315-332Publisher:
- Savez farmaceutskih udruženja Srbije, Beograd
Collections
Institution/Community
PharmacyTY - JOUR AU - Đurić, Zorica AU - Jovanović, Milica AU - Parojčić, Jelena AU - Ibrić, Svetlana PY - 2004 UR - https://farfar.pharmacy.bg.ac.rs/handle/123456789/491 AB - In this report preparations of laxatives and antidiarrhoeals and the technological procedures used in production, have been reviewed.The importance of special technological procedure as freeze drying in the production and stabilisation has been explained. The most frequent dosage forms for these drugs are tablets.Good physical characteristics of tablets, insignificant variation of drug content, uniformity of dosage as required bioavailability are to bi provided by using adequate combination of excipients in the formulation and by proper selection of production method and order of technological operations.Additional requirements are to be achieved in the production of chewable tablets , frequently used as a dosage form for laxatives as calcium polycarbophil. Basic concept of tablet production validation is included in this report. AB - U radu su prikazani lekoviti preparati laksativa i antidijaroika i metode koje se koriste u proizvodnji. Objašnjen je značaj specijalnih tehnoloških postupaka kao što je liofilizacija u proizvodnji i stabilizaciji nekih proizvoda iz ove grupe.Najčešće primenjivani oblik ovih lekovitih supstanci su tablete. Za proizvodnju tableta koje će imati dobre fizičke karakteristike, zanemarljivo mala odstupanja u sadržaju leka, jednolikost doze kao i potrebnu bioraspoloživost, koristi se adekvatna kombinacija pomoćnih materija u formulaciji i pravilan izbor metode izrade. Dodatni zahtevi se postavljaju u slučaju proizvodnje tableta za žvakanje, kao što su tablete sa kalcijum polikarbofilom. U radu su dati i osnovni principi validacije procesa proizvodnje tableta. PB - Savez farmaceutskih udruženja Srbije, Beograd T2 - Arhiv za farmaciju T1 - Preparations of laxatives and antidiarrhoeals: Pharmaceutically - technological aspect T1 - Lekoviti preparati lakasativa i antidijaroika - farmaceutsko tehnološki aspekt VL - 54 IS - 3 SP - 315 EP - 332 UR - https://hdl.handle.net/21.15107/rcub_farfar_491 ER -
@article{ author = "Đurić, Zorica and Jovanović, Milica and Parojčić, Jelena and Ibrić, Svetlana", year = "2004", abstract = "In this report preparations of laxatives and antidiarrhoeals and the technological procedures used in production, have been reviewed.The importance of special technological procedure as freeze drying in the production and stabilisation has been explained. The most frequent dosage forms for these drugs are tablets.Good physical characteristics of tablets, insignificant variation of drug content, uniformity of dosage as required bioavailability are to bi provided by using adequate combination of excipients in the formulation and by proper selection of production method and order of technological operations.Additional requirements are to be achieved in the production of chewable tablets , frequently used as a dosage form for laxatives as calcium polycarbophil. Basic concept of tablet production validation is included in this report., U radu su prikazani lekoviti preparati laksativa i antidijaroika i metode koje se koriste u proizvodnji. Objašnjen je značaj specijalnih tehnoloških postupaka kao što je liofilizacija u proizvodnji i stabilizaciji nekih proizvoda iz ove grupe.Najčešće primenjivani oblik ovih lekovitih supstanci su tablete. Za proizvodnju tableta koje će imati dobre fizičke karakteristike, zanemarljivo mala odstupanja u sadržaju leka, jednolikost doze kao i potrebnu bioraspoloživost, koristi se adekvatna kombinacija pomoćnih materija u formulaciji i pravilan izbor metode izrade. Dodatni zahtevi se postavljaju u slučaju proizvodnje tableta za žvakanje, kao što su tablete sa kalcijum polikarbofilom. U radu su dati i osnovni principi validacije procesa proizvodnje tableta.", publisher = "Savez farmaceutskih udruženja Srbije, Beograd", journal = "Arhiv za farmaciju", title = "Preparations of laxatives and antidiarrhoeals: Pharmaceutically - technological aspect, Lekoviti preparati lakasativa i antidijaroika - farmaceutsko tehnološki aspekt", volume = "54", number = "3", pages = "315-332", url = "https://hdl.handle.net/21.15107/rcub_farfar_491" }
Đurić, Z., Jovanović, M., Parojčić, J.,& Ibrić, S.. (2004). Preparations of laxatives and antidiarrhoeals: Pharmaceutically - technological aspect. in Arhiv za farmaciju Savez farmaceutskih udruženja Srbije, Beograd., 54(3), 315-332. https://hdl.handle.net/21.15107/rcub_farfar_491
Đurić Z, Jovanović M, Parojčić J, Ibrić S. Preparations of laxatives and antidiarrhoeals: Pharmaceutically - technological aspect. in Arhiv za farmaciju. 2004;54(3):315-332. https://hdl.handle.net/21.15107/rcub_farfar_491 .
Đurić, Zorica, Jovanović, Milica, Parojčić, Jelena, Ibrić, Svetlana, "Preparations of laxatives and antidiarrhoeals: Pharmaceutically - technological aspect" in Arhiv za farmaciju, 54, no. 3 (2004):315-332, https://hdl.handle.net/21.15107/rcub_farfar_491 .